Why is buprenorphine less addictive than other opioids

Why is buprenorphine less addictive than other opioids (such as fentanyl) - is it understandable by its strength of binding to the general receptor?

E

Expert

Verified

Buprenorphine is what is termed to as a partial agonist; that is, it binds to the receptor however even at its maximum can’t provide as much of an effect as a full agonist (like morphine) - it is, therefore, as well a partial antagonist (partly inhibits the actions of full agonists).

As addiction is probable to be linked to strength of the consequence of the drug, buprenorphine has much less effect and, thus, less addiction.

   Related Questions in Biology

  • Q : Needs and Goals - Motivation -

    Both are interdependent; neither exists without the other. However, people are often not as aware of their needs as they are of their goals. For example, a teenager may not consciously be aware of his social needs but may join a photography club to meet new friends. A loc

  • Q : Main endocrine functions of the placenta

    What are the main endocrine functions of the placenta?

  • Q : Type of plant tissue is cork State type

    State type of plant tissue is cork?

  • Q : Types | Channels of Communication -

    Communication in an organization carries innumerable kinds of messages which may be difficult to map out; but it may be possible to classify communications in regard to how to transmit. Or who communicates to whom, or what kinds of relationships communication develop. Thus, communication may be g

  • Q : What is parthenogenesis What is meant

    What is meant by the parthenogenesis?

  • Q : What is SAP R-3 SAP R/3 : It is a third

    SAP R/3: It is a third generation set of highly integrated software modules which executes common business function mainly based on multinational leading practice. Takes care of any venture though diverse in operation, spread over the globe. In R/3 sy

  • Q : Modes of transmission-main

    Write down the modes of transmission, main signs and treatments and symptoms of hepatitis B?

  • Q : Face to Face Communication -

    This type of communication may, at the first thought, appear to be identical with oral communication. However, it is possible to visualize certain situation on which the two get distinguished. Telephonic conversation is oral but we cannot call it face-to dace communication. the presidents of two

  • Q : Examples of secretory cells What are

    What are various examples of secretory cells?

  • Q : Explanation of hypersensitive reactions

    Give a brief explanation of hypersensitive reactions.

©TutorsGlobe All rights reserved 2022-2023.